CC-115 (CC115) is a novel and potent dual inhibitor of DNA-PK (DNA-dependent protein kinase) and mTOR (mammalian target of rapamycin) with IC50s of 13 nM and 21 nM, respectively and with potential antineoplastic activity.

ME0328 (ME-0328) is a novel, potent and selective inhibitor of Poly (ADP-ribose) polymerase (PARP) with potential anticancer activity.

AZD-5305 (AZD5305) is a novel, potent, selective and orally bioactive PARP [Poly(ADP-ribose)polymerase-1] inhibitor with anticancer activity.

Pamiparib maleate, the maleate salt of pamiparib (formerly BGB-290), is a selective inhibitor of PARP1 and PARP2 with IC50 values of 0.83 and 0.11 nM, respectively.

BGP-15 is a potent PARP inhibitor that can protect against heart failure and atrial fibrillation in mice.

RHPS4 methosulfate (also known as NSC714187) is a potent inhibitor of telomerase with submicromolar activity.

Quinine HCl dihydrate (Quinine hydrochloride dihydrate) is a novel, potent naturally occuring compound with a variety of biological activities such as anti-malarial, antipyretic, analgesic , anti-inflammatory properties.

Psoralen (psoralene, Ficusin, Furocoumarin) is a naturally occurring furocoumarin isolated from Fructus Psoraleae, it intercalates with DNA, inhibiting DNA synthesis and cell division.

Rucaparib (formerly known as AG-14447; AG-014699; PF-01367338; Rubraca) is an inhibitor of PARP [ (poly(ADP-Ribose) polymerase)] with anticancer effects.

Niraparib R-enantiomer, the R-isomer of Niraparib, is a potent PARP1 [poly(ADP-Ribose) polymerase] inhibitor (IC50 = 2.4 nM) with anticancer activity.