AMG 333 is a novel, potent and highly selective TRPM8 antagonist with an IC50 of 13 nM and 20 nM for hTRPM8 and rTRPM8, respectively.

ML-SA1 is a potent agonist of TRPML1 (transient receptor potential mucolipin 1) with broad spectrum of antiviral activity.

TRPV4 agonist (no formal name), is a novel and potent agonist of TRPV4 with EC50 of 60 nM in the hTRPV4 Ca2+ assay

Trovafloxacin mesylate (CP-99219) is a broad-spectrum quinolone antibiotic that inhibits DNA supercoiling in various bacteria by blocking the activity of DNA gyrase and topoisomerase IV.

Beta-Eudesmol is a novel and potent oxygenated sesquiterpene.

Pyr6 is a novel, potent, selective and pyrazole-based inhibitor of Ca2+ entry mediated by transient receptor potential cation 3 (TRPC3) channels.

GSK2193874 (GSK-2193874) is a novel, potent, orally bioactive, and selective TRPV4 (Transient Receptor Potential Vanilloid 4) antagonist with the potential to be used for congestive heart failure.

Nonivamide is a novel and potent capsaicin analogue.

ML SI3 (ML-SI3) is an antagonist of the TRPML family of calcium channels.

TRPV4 agonist-1 free base is a novel and potent transient receptor potential vanilloid 4 (TRPV4) agonist .