ZLDI-8 is a novel and potent enzyme ADAM-17 inhibitor
Tamoxifen-d5 is a penta-deuterated form of Tamoxifen (ICI 47699), which is an anticancer drug and a selective estrogen receptor modulator (SERM).
Carveol is a novel and potent endogenous metabolite
Heraclenin is a novel and potent polyacetylene
4-Methylherniarin is a novel and potent coumarin analogue
JPI-547 HCl, dual inhibitor of PARP1/2 and TNKS1/2
Cortistatin-14 TFA (CST-14) is a novel and potent cyclic neuropeptide that has structural similarity to somatostatin-14. Cortistatin-14 exerts anticonvulsive, neuroprotective effect and anti-inflammatory activity by binding to the somatostatin receptors (sst1-sst5). Cortistatin (CST-14) is a recently discovered endogenous peptide which shares similarity to somatostatin and binds to somatostatin receptors.
Latanoprost lactone diol is an intermediate used in the synthesis of Latanoprost, which is a FP receptor agonist (EC50 = 3.6 nM for human FP receptors) with the potential for the treatment of glaucoma.
HSV-TK substrate is a novel and potent substrate for HSV-TK
2,3,4,5-Tetracaffeoyl-D-Glucaric acid is a novel and potent caffeoyl-D-glucaric acid analogue