α-Lipoic Acid (Thioctic acid; (±)-α-Lipoic acid; DL-α-Lipoic acid) is a novel organosulfur compound which acts as an antioxidant, and is an essential cofactor of mitochondrial enzyme complexes.

Caffeic acid phenethyl ester (also called CAPE; BAF-IN-C09; 2-Phenylethyl Caffeate; β-Phenylethyl Caffeate), a naturally occuring compound isolated from honeybee hive propolis, is potent and specific inhibitor of NF-κB activation with antioxidant, anticancer, immunomodulatory and antiinflammatory activities.

Andrographolide, a naturally occuring labdane diterpenoid extracted from the stem and leaves of Andrographis paniculata, is an irreversible/covalent NF-κB inhibitor with potential anti-inflammatory activity.

Barlerin is a novel and potent iridoid glucoside.

Laquinimod (also known as ABR-215062, LAQ) is a potent and orally bioactive immunoregulator being investigated for treatment of multiple sclerosis (MS).

JSH-23 HCl is designed as an inhibitor of NF-κB transcriptional activity with IC50 of 7.1 μM in RAW 264.7 cell line.

Berbamine 2HCl is a naturally occuring isoquinoline alkaloid found in traditional Chinese medicine Barberry with anti-tumor, immunomodulatory and cardiovascular effects.

Enzymatically modified isoquercitrin, formerly known as EMIQ, is a flavonoid.

Ophiopogonin D is a novel and potent C29 steroidal glycoside.

Zingerone is a novel and potent anti-inflammatory, antidiabetic, antilipolytic, antidiarrheal, and antispasmodic compound.