Bisoprolol fumarate (Zebeta; (+/-)-Bisoprolol hemifumarate; Bisobloc; EMD 33512; EMD33512), the fumarate salt of bisoprolol, is a potent and selective β1 adrenergic receptor antagonist/blocker with potential antihypertensive and cardioprotective activities.

Rucaparib CAMSYLATE (AG014699; AG14447; PF01367338; trade name: Rubraca), the CAMSYLATE salt of rucaparib, is a potent PARP inhibitor approved by FDA for the treatment of ovarian cancer.

GA 017 is a novel,potent and selective inhibitor of LATS1 and LATS2 (large tumor suppressor kinase 1/2).

TAK-441 is a novel, orally bioavailable, potent and selective Hedgehog (Hh) signaling pathway inhibitor with acceptable solubility and pharmacokinetic properties.

BDA-366 (BDA366) is a potent and selective small-molecule antagonist of the Bcl2-BH4 domain with potential anticancer activity.