Gpi-688, glycogen phosphorylase (GPa) inhibitor

Apraclonidine (iopidine) is a novel and potent α2 receptor agonist used in glaucoma therapy. It is also a weak alpha-1 adrenergic receptor agonist. Apraclonidine enhances aqueous humor uveoscleral outflow and decreases aqueous production by vasoconstriction.

TP748 is a novel and potent isoxazole

Harmol is a natural chemical compound classified as a β-carboline. It is readily formed in vivo in humans by O-demethylation of harmine.

(R)-NVS-ZP7-4 is a novel and potent Zinc transporter SLC39A7 (ZIP7) inhibitor

Besifloxacin is a novel and potent fluoroquinolone antibiotic agent

SIAIS178 is a novel and potent BCR-ABL degrader

HIF-1/2α-IN-2, inhibitor of HIF-1/2α

Piperaquine, antimalarial drug

GSK-2793660 is a novel and potent inhibitor of Cathepsin C (CTSC)