Luteolin 7-O-glucuronide could inhibit Matrix Metalloproteinases (MMP) activities, with IC50s of 17.63, 7.99, 11.42, 12.85, 0.03 μM for MMP-1, MMP-3, MMP-8, MMP-9, MMP-13, respectively.

Phosphoramidon disodium salt is a potent metalloendopeptidase inhibitor, which is widely used as a biochemical research tool.

20(R)-Ginsenoside Rh2 is a novel and potent matrix metalloproteinase (MMP) inhibitor.

GW280264X is a novel and potent ADAM17 inhibitor.

Histatin 5 is a novel and potent bioactive peptide compound that inhibits the activity of MMP-2 and MMP-9 (host matrix metalloproteinases ) with IC50s of 0.57 and 0.25 μM, respectively.

CTS-1027 is a novel, potent small molecule inhibitor of MMPs (matrix metalloproteinase) with IC50s of 0.3 nM, 0.5 nM for MMP2, MMP13, respectively, and has > 1,000 fold selectivity over MMP1.