Bromocriptine Mesylate (CB154) is a dopamine D2/3 agonist (with pKi of 8.05±0.2 for D2) for the treatment of pituitary tumors, Parkinson’s disease (PD), hyperprolactinaemia, neuroleptic malignant syndrome, and type 2 diabetes.
Dopamine HCl (formerly Intropin; Dopamine HCl; ASL 279; ASL279; P 498; 3-Hydroxytyramine, ASL-279 and Intropin), the hydrochloride salt of dopamine, is an endogenous catecholamine neurotransmitter found in a wide variety of animals, it is a dopamine D1-5 receptors agonist.
FAUC 346 is a novel , potent and highly selective D3 partial agonist .
Cariprazine HCl (formerly MP-214; RGH-188; MP214; RGH188; Vraylar; Reagila), the hydrochloride salt of cariprazine, is an antipsychotic medication that has been approved for the treatment of schizophrenia, as well as for bipolar disorder (manic/mixed and depressive episodes), and as an adjunctive agent for the treatment of major depressive disorder.
Pimozide (R-6238; NSC-170984; Orap) is an antipsychotic drug of the diphenylbutylpiperidine class discovered y Janssen Pharmaceuticals in 1963.
Haloperidol (R1625; Eukystol; HSDB-3093; Haldol; Serenace; Aloperidin) is a potent antipsychotic medication acting as a dopamine D2 receptor antagonist.
Dexpramipexole (also known as KNS-760704, R-(+)-Pramipexole and (R)-Pramipexole), an enantiomer of pramipexole, is a dopamine agonist of the non-ergoline class with the potential for the treatment of amyotrophic lateral sclerosis (ALS) (also known as Lou Gehrig’s disease).
SKF-82958 HBr, the hydrobromide salt of SKF-81297, is a novel, potent and selective dopamine D1/D5 receptor full agonist which stimulates motor behaviour of MPTP-lesioned monkeys.
SCH-23390 is a potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types, respectively).
Amfebutamone HCl (Bupropion, Wellbutrin, Zyban; BW-323; NSC315851; NSC-315851), the hydrochloride salt of Amfebutamone, is a potent and selective norepinephrine-dopamine reuptake inhibitor used as an antidepressant and for smoking cessation.