Rocuronium Bromide (ORG-9426; Zemuron; Esmeron; Esmeron; Esmerone) is a potent and competitive Nicotinic acetyl-choline receptors (AchR) antagonist, which is a non-depolarizing neuromuscular blocking agent used in anaesthesia required for surgery or mechanical ventilation.

Isoimperatorin is a COX-2 inhibitor.

PNU-120596 (PNU120596; NSC 216666; PNU 120596; NSC-216666) is a potent and selective PAM (positive allosteric modulator) of α7 nAChR (acetylcholine receptor) with an EC50 of 216 NM.

Diphenidol HCl (Vontrol; Difenidol), the hydrochloride salt of diphenidol which is an antiemetic, is a potent antagonist of muscarinic M2 and M3 receptors used as an antiemetic and as an antivertigo agent.

Pyridostigmine Bromide (Mestinon; Regonol; Kalimin) is a parasympathomimetic and a reversible cholinesterase inhibitor used in the treatment of myasthenia gravis and to reverse the actions of muscle relaxants. Pyridostigmine Bromide hase been approved for millitary use during the Gulf War as a pretreatment to protect troops from the harmful effects of nerve agents.

Pancuronium dibromide (OrgNA97; NA-97; Org NA 97; Pavulon), a neuromuscular relaxant used in euthanasia, is a bis-quaternary steroid and a competitive nicotinic acetylcholine receptor antagonist with an IC50 of 5.5 nM.

Neostigmine Bromide (Eustigmin bromide; Neoserine bromide) is a reversible acetylcholinesterase inhibitor and a medication used to treat myasthenia gravis, Ogilvie syndrome, and urinary retention without the presence of a blockage.

Sulfoxaflor (GF-2372; XDE-208) is a sulfoximine-based systemic insecticide which acts as an agonist of nAChR1 and nAChR2.

Paroxetine HCl (formerly BRL-29060A, BRL29060A, FG7051; FG-7051), the hydrochloride salt of Paroxetine, is a potent and selective serotonin uptake inhibitor (SSRI) that is effective in the treatment of depression.

Butylscopolamine bromide is a potent antimuscarinic quaternary ammonium analogue acting as a competitive antagonist of mAChR (IC50: 55.3 ± 4.3 nM).