Dichloroacetate (CPC-211; DCA; X-11S) is a potent and specific inhibitor of pyruvate dehydrogenase kinase (PDK) with IC50 values of 183 and 80 μM for PDK2 and PDK4 respectively.

Neohesperidin dihydrochalcone (Neohesperidin DC; NHDC), an artificial sweetener and a synthetic glycoside chalcone, is added to various foods and beverages as a low caloric artificial sweetener.

NXY-059 (also known as Cerovive, OKN007, Disufenton Sodium) is a disulfonyl derivative that has shown a significant differences in arterial Po2 and pH between the experimental groups before ischemia in BBB permeability study with Po2 value of 112.9±9.7mm Hg and pH value of 7.443±0.01.

Procyanidin B2 is a novel and potent flavanoid.

DMNQ is a superoxide generating agent.

OBA-09 (OBA09) is a novel and potent neuroprotective agent.

Coelenterazine, a luciferin which is a light-emitting molecule, is a luminescent enzyme substrate that is used for monitoring reporter genes in BRET, ELISA and HTS techniques.

Calycosin-7-O-β-D-glucoside is a novel and potent melanin biosynthesis inhibitor.

CADD522 is a novel and potent inhibitor of runt-related transcription factor-2 (RUNX2)-DNA binding with an IC50 of 10 nM.

Norbergenin( Demethylbergenin) is the O-demethyl derivative of bergenin.