S-Bimanylcysteine is a novel and potent bioactive compound

ACG-548B is a potent, selective choline kinase α (ChoKα) inhibitor.

Atpenin A5 is a novel and potent inhibitor of IGF-IR

Clobenzorex has been discontinued (DEA controlled substance). Clobenzorex is an optically active N-substituted analogue of (+)amphetamine.

Terizidone (Terivalidin), a derivate of cycloserine (CS), is a bacteriostatic second-line drug for multi-drug-resistant tuberculosis (MDR-TB) in conjunction with other second-line drugs. It is used internationally, but is not currently approved in the United States. It is a combination of two molecules of CS. The MOA includes competitively inhibiting l-alanine racemase and d-alanine ligase to […]

Ancarolol is a novel and potent beta blocker

Retroprogesterone is a novel and potent progestin

Ro 24-0238 is a novel and potent platelet-activating factor-antagonist

BAYu9773 is a novel and potent CysLT1 and CysLT2 receptor antagonist

MK-386 is a novel, potent and selective human type-1 5alpha-reductase inhibitor.