MDL-29951 is a potent glycine antagonist of NMDA (N-methyl-D-aspartate) receptor activation with Ki value of 0.14 μM in an in vitro and in vivo [3H]glycine binding assay.

ZL006 is an efficient inhibitor of the nNOS/PSD-95 protein-protein interaction and showed great promise in cellular experiments and animal models of ischemic stroke and pain.

PhTx-74 HCl (Philanthotoxin 74; PhTx 74; PhTx74), the dihydrochloride salt of PhTx-74, is an analogue of philanthotoxin-4,3,3 which is a naturally-occurring wasp venom toxin.

GNE-8324 (GNE8324) is a novel, potent and selective PAM (Positive Allosteric Modulators) of NMDA receptor. NMDA Receptors (NMDARs) play key roles in synaptic physiology and NMDAR hypofunction has been implicated in various neurological conditions.

Eliprodil (formerly known as SL-820715) is a non-competitive NR2B-NMDA receptor antagonist with IC50 value of 1 uM, it is less potent for NR2A- and NR2C-containing receptors with IC50 > 100 uM.

Sepimostate mesilate(also known as FUT-187or TO 187) is an inhibitor used in therapy of pancreatitis, it inhibits the Ifenprodil binding with a Ki value of 27.7 µM.

PEPA is a novel and potent modulator of AMPA receptors.