Ethisterone (Aethisteron; Progestoral; NSC-9565; NSC9565) is a progestogen hormone and a synthetic contraceptive that is being developed as an anticancer agent for the treatment of prostate cancer.
Bazedoxifene HCl (formerly TSE-424; WAY-140424; WAY140424; TSE424; Viviant), the hydrochloride salt of Bazedoxifene, is a non-steroidal, indole-based and 3rd generation selective estrogen receptor modulator (SERM) with potential antineoplastic activity.
Mestranol (Ethinyl Estradiol 3 Methyl Ether; Devocin; Norquen; Ovastol), the 3-methyl ether of ethinyl estradiol, is a potent estrogen receptor agonist that has been used as an oral contraceptive.
Progesterone (Pregn-4-ene-3,20-dione; Hormoflaveine; Lutociclina; Agolutin; Crinone; Luteohormone; Utrogestan; Cyclogest) is an endogenous steroidal hormone and a universal precursor for the biosynthesis of other steroidal hormones.
Gestodene (WL-70, Δ15-norgestrel or 15-dehydronorgestrel; Gestodeno; Gestodenum; Gestoden; Gestodene; Gestodene, SHB 331; SHB-331;WL-70; SHB 331; WL 70; SHB331; WL70) is a potent progestogen hormonal contraceptive.
Medroxyprogesterone acetate (formerly NSC26386; NSC 26386; Medroxyprogesterone 17-acetate; MPA), the 17-ester form of Medroxyprogesterone, is a steroidal progestin and a synthetic variant of the human hormone progesterone.
Tariquidar dimesylate (formerly known as XR9576; D06008; XR-9576; D-06008), the dimesylate salt of Tariquidar, is a novel potent and selective noncompetitive inhibitor of P-glycoprotein (P-gp) with potential antitumor activity.
Altrenogest (also known as Allyltrenbolone; A35957; RU2267; DRC6246; R-2267; A-35957; RU-2267; Allyl trenbolone; REGU-MATE; Regumate) is a progestogen structurally related to veterinary steroid trenbolone.
Bazedoxifene acetate (formerly TSE-424; WAY140424; WAY-140424; TSE424; Viviant), the acetic acid salt form of Bazedoxifene, is a 3rd generation selective estrogen receptor modulator (SERM) with IC50s of 26 and 99 nM for ERα and ERβ, respectively.
Estriol (also called NSC12169; NSC 12169; NSC-12169; Oestriol) is a potent antagonist of the G-protein coupled estrogen receptor in estrogen receptor-negative breast cancer cells.