Nimodipine (formerly BAY E 9736; BAY-E-9736, Nimotop, Periplum) is a potent dihydropyridine/DHP class of calcium channel blocker (CCB) and an autophagy inhibitor with antihypertensive effects.

Dioscin (CCRIS 4123; Collettiside III) is a naturally occuring saponin isolated from Polygonatum Zanlanscianense Pamp, showing antitumor activities.

CA-5f (CA5f) is a novel and potent late-stage macroautophagy/autophagy inhibitor via inhibiting autophagosome-lysosome fusion with anti-tumor activity.

Valproic acid is an HDAC (Histone deacetylase) inhibitor used in the treatment of epilepsy, bipolar disorder and prevention of migraine headaches.

Temozolomide (Methazolastone; CCRG81045; NSC 362856; SCH 52365; MB39831; and RP46161) is an orally bioavailable and brain penetrant DNA alkylating agent / damage inducer used as an anticancer drug.

TFEB activator 1 is a potent, orally bioactive, and mTOR-independent activator of TFEB with neuroprotective effects.

AS1842856 is a novel potent, orally active and cell-permeable small-molecule inhibitor of Foxo1 (forkhead transcription factor forkhead box O1) with an IC50 of 30 nM.

5-Aminolevulinic acid HCl (also known as ALA hydrochloride; trade name: Levulan), an FDA approved drug for treating actinic keratosis, is an intermediate in heme biosynthesis and the universal precursor of tetrapyrroles.

Lys05, or Lys01 trihydrochloride, is a potent, water soluble lysosomal autophagy inhibitor.

Vinorelbine (KW-2307; Nor-5′-anhydrovinblastine) is a potent antimitotic agent and a semisynthetic vinca alkaloid derived from the leaves of the periwinkle plant (Vinca rosea) used for the treatment for some types of cancer, including breast cancer and non-small cell lung cancer.