A2764 diHCl
This product is for research use only, not for human use. We do not sell to patients.
For small sizes, please check our retail website as below: www.invivochem.com
| Size | Price | Stock |
|---|---|---|
| 500mg | $950 | Check With Us |
| 1g | $1350 | Check With Us |
| 5g | $3645 | Check With Us |
: Cat #: V37830 CAS #: 861038-72-4 Purity ≥ 98%
Description: A2764 diHCl is a novel and potent inhibitor of TRESK.
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| Molecular Weight (MW) | 351.70 |
|---|---|
| Molecular Formula | C₁₅H₂₁Cl₃N₂O |
| CAS No. | 861038-72-4 |
| Synonyms | A 2764 diHCl |
| Protocol | In Vitro | A2764 (100 µM) shows an improved inhibitory potency for activated channel with an IC50 of activated channel in ionomycin-activated mTRESK current.The subsequent application of A2764 strongly inhibits the current (77.8±3.5%) |
|---|
These protocols are for reference only. InvivoChem does not
independently validate these methods.
| Solvent volume to be added | Mass (the weight of a compound) | |||
|---|---|---|---|---|
| Mother liquor concentration | 1mg | 5mg | 10mg | 20mg |
| 1mM | 2.8433 mL | 14.2167 mL | 28.4333 mL | 56.8666 mL |
| 5mM | 0.5687 mL | 2.8433 mL | 5.6867 mL | 11.3733 mL |
| 10mM | 0.2843 mL | 1.4217 mL | 2.8433 mL | 5.6867 mL |
| 20mM | 0.1422 mL | 0.7108 mL | 1.4217 mL | 2.8433 mL |
The molarity calculator equation
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The dilution calculator equation
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This equation is commonly abbreviated as: C1 V1 = C2 V2
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Step One: Enter information below
Dosage mg/kg
Average weight of animals g
Dosing volume per animal µL
Number of animals
Step Two: Enter the in vivo formulation
%DMSO
+
%
+
%Tween 80
+
%ddH2O
Calculation Results:
Working concentration:
mg/ml;
Method for preparing DMSO master liquid:
mg
drug pre-dissolved in
µL
DMSO(Master liquid concentration
mg/mL)
,Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.
Method for preparing in vivo formulation:
Take
µL
DMSO master liquid, next add
µL
PEG300, mix and clarify, next add
µL
Tween 80,mix and clarify, next add
µL
ddH2O,mix and clarify.
Note:
- (1) Please be sure that the solution is clear before the addition of next solvent. Dissolution methods like vortex, ultrasound or warming and heat may be used to aid dissolving.
- (2) Be sure to add the solvent(s) in order.