K-Ras(G12C) inhibitor 12 is a co-valent and allosteric inhibitor of K-Ras G12C with potential antitumor activity.

CCG-100602 is a novel and potent bioactive compound.

EHT 1864 2HCl (EHT-1864; EHT1864), the dihydrochloride salt of EHT-1864, is a potent and novel Rac family GTPase inhibitor with important biological activity.

6H05 TFA (6H-05; 6 H05), the trifluoroacetic acd salt of 6H05, is a potent, covalent, selective and allosteric inhibitor of K-Ras (G12C) which is oncogenic.

Zoledronic acid (Zoledronate; CGP-42446; CGP42446A; ZOL-446; Zometa; Reclast) is potent bisphosphonate with anti-bone-resorption activity.

MLS-573151 is a novel, specific, cell permeable inhibitor of Cdc42 (IC50 = 2 μM).

NSC 23766 (NSC-23766; NSC23766) is a novel, selective and potent inhibitor of Rac GTPase with anti-influenza virus activity.

Salirasib (known also as S-Farnesylthiosalicylic acid; Farnesyl Thiosalicylic Acid; FTS), a salicylic acid analog, is a potent and competitive prenylated protein methyltransferase (PPMTase) inhibitor with potential antineoplastic activity.

CCG-1423 (CCG1423; CCG 1423) is a novel, potent and specific small-molecule inhibitor of RhoA signaling pathway with potential antitumor activity.