Mevastatin (CS500; ML236B; Mevastatin; Compactin; ML-236B), an approved anti-hyperliperdemic drug of the statin class, is a potent and competitive inhibitor of HMG-Coenzyme A (HMG-CoA) reductase with anti-hyperlipidemic effects.

Rosuvastatin Calcium (S-4522, Rosuvastatin hemicalcium; ZD-4522; ZD4522, trade name: Crestor), a member of the statin class of lipid-lowering drugs, is a potent and competitive inhibitor of HMG-CoA reductase with potential anti-hyperlipidemic activity.

Lovastatin (Mevinolin; Mevacor; MK-803; Altoprev; Monacolin K; MK803), belonging to the statin class of hypolipidemic agent/lipid-lowering drugs, is a potent and cell-permeable inhibitor of HMG-CoA reductase with potential anti-hyperlipidemic effects.

Rosuvastatin (S-4522; ZD-4522; S4522; ZD4522; trade name: Crestor) is a member of the statin class of antihyperlipidemic drugs which acts as a competitive inhibitor of HMG-CoA reductase with IC50 of 11 nM in a cell-free assay.

Clinofibrate (Lipoclin; S-8527; S 8527) is a potent anti-hyperlipidemic agent which acts as an HMG-CoA (hydroxymethylglutaryl coenzyme A) reductase inhibitor with potential anti-hyperlipidemic effects.

Pravastatin sodium (Apotex; CS-514; Pravachol; Pravaselect; Apo-Pravastatin; Mevalotin; Elisor; Lipostat), an approved hypolipidemic drug of the statin class, is an HMG-CoA reductase inhibitor against sterol synthesis with potential anti-hyperlipidemic effects.

Atorvastatin Calcium (Lipitor; CI-981; CI981; Atorvastatin hemicalcium; liptonorm), an approved blockbuster drug of the statin class of LDL cholesterol-lowering/hypolipidemic medications, is a potent and selective inhibitor of HMG-CoA reductase with anti-hyperlipidemic effects.

Fluvastatin (XU-62320; Fluindostatin; Lescol XL; XU-62-320; Canef; Lipaxan; Vastin), an approved drug belonging to the statin class of hypolipidemic medications, is a potent inhibitor of HMG-CoA reductase activity with potential anti-hyperlipidemic effects.

Rosuvastatin D3 Sodium is deuterium labeled Rosuvastatin (also known as S-4522 and ZD 4522, trade name: Crestor) which is a member of the statin class of drugs and a competitive inhibitor of HMG-CoA reductase with IC50 of 11 nM in a cell-free assay.

Rosuvastatin D6 Calcium is deuterium labeled Rosuvastatin Calcium (also known as S-4522, Rosuvastatin hemicalcium; ZD 4522 Calcium and ZD 4522, trade name: Crestor) which is a member of the statin class of drugs and a competitive inhibitor of HMG-CoA reductase with IC50 of 11 nM in a cell-free assay.