Fipronil is a phenylpyrazole-based insecticide with a broad-spectrum insecticidal activity.

Bemegride (3-Ethyl-3-methylglutarimide; Antibarbi; Agipnon; Ahypnon; Eukraton; Malysol; Mikedimide; Zentraleptin) is apotent central nervous system stimulant and effective antidote for barbiturate poisoning.

Cgp 52432 is a novel and highly potent GABA-B receptor antagonist with an IC50 of 85 nM.

(-)-Bicuculline methochloride (l-Bicuculline methochloride), an enantiomer of (+)-bicuculline methochloride, is a highly potent GABAA receptor antagonist.

Nifedipine (Adalat, Procardia, Bay-1040, BAY-a-1040; Cordipin, Corinfar, Bay 1040) is a dihydropyridine calcium channel blocker (CCB) with antihypertensive effects.

Dihydromyricetin (also known as Ampelopsin, Ampeloptin, DHM) is a naturally occuring flavonoid isolated from Ampelopsis grossedentata with antioxidant activity.

L-cycloserine is an irreversible inhibitor of the GABA pyridoxal 5′-phosphate-dependent aminitransferase in E. coli, as well in the brains of various animals.

AZD-6280 is a novel, potent and selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder.

Ginkgolide A (Ginkgolide A; BN 52020; BN-52020), a naturally occuring terpenic lactone isolated from Ginkgo biloba, is a g-aminobutyric acid (GABA) receptor antagonist with important biological activity.

Guvacine HCl, the hydrochloride salt of Guvacine, is an alkaloid isolated from the nut of Areca catechu which acts as an inhibitor of GABA transporter, and dispalys modest selectivity for cloned GABA transporters with IC50s of 14 μM (human GAT-1), 39 μM (rat GAT-1), 58 μM (rat GAT-2), 119 μM (human GAT-3), 378 μM (rat […]