Praeruptorin B, a naturally occuring compound from roots of Peucedanum praeruptorum Dunn, is a potent inhibitor of sterol regulatory element-binding proteins (SREBPs).

FT113 is a potent and orally bioavailable fatty acid synthase (FASN) inhibitor, with an IC50 of 213 nM for full-length recombinant human FASN enzyme.

Desoxyrhaponticin is a novel and potent stilbene glycoside from the Tibetan nutritional food Rheum tanguticum Maxim.

PF429242 dihydrochloride is a novel, potent, reversible and competitive S1P [sterol regulatory element-binding protein (SREBP) site 1 protease] inhibitor with an IC50 of 170 nM.

Lycorine is a novel and potent inhibitor of the growth and metastasis of hormone-refractory prostate.

GSK2194069 is a novel, potent and specific inhibitor of the β-ketoacyl reductase (KR) activity of hFAS with an IC50 of 7.7 ± 4.1 nM in an assay detecting released CoA.

C75 trans [(±)-C75] is an isomer/enantiomer of C75 which is a synthetic fatty-acid synthase (FASN) inhibitor.

Fatostatin hydrochloride is a novel and potent inhibitor of SREBP.

FGH10019 is a novel and potent inhibitor of the sterol regulatory element-binding protein (SREBP) with IC50 of 1 μM.