T16Ainh-A01 is an aminophenylthiazole analog acting as a novel and potent transmembrane protein 16A (TMEM16A) inhibitor which inhibits TMEM16A-mediated chloride currents with an IC50 value of ~1 µM.

Shikonin (C.I. 75535; Isoarnebin 4) is a natural product and major component of the Chinese medicin ‘zicao’ with various biological activities such as anti-inflammatory activity by inhibition of TNF-α, NF-κB, HIV-1.

Talniflumate (BA -602-06), a prodrug of Niflumic acid, is a potent,orally bioactive and selective inhibitor of core mucin-synthesizing enzyme GCNT3 (core 2b-1,6 N-acetylglucosaminyltrans-ferase).

CaCCinh-A01 (also known as TMEM16 Blocker I) is an inhibitor of TMEM16A and calcium-activated chloride channel (CaCC) with IC50s of 2.1 and 10 μM, respectively.

Ani9 is a novel and potent ANO1 inhibitor.

NS1652 is a novel, reversible anion conductance inhibitor which blocks chloride channel with an IC50 of 1.6 μM in human and mouse red blood cells.