Pralidoxime Chloride (2-PAM chloride) is a useful anti-dote agent for organophosphate poisoning.

Violanthin is a naturally occuring flavanoid 8-c-glycoside acting as a potent acetylcholinesterase (AChE) inhibitor with IC50 of 79.80 μM.

Scopoletin (Gelseminic acid; Chrysatropic acid) is a naturally occurring coumarin acting as an inhibitor of acetylcholinesterase (AChE), has anti-hyperuricemic effect.

Epiberberine Chloride, an alkaloid, is a natural anticancer agent isolated from Coptis chinensis with the potential for the treatment of diabetic disease., it acts as a potent AChE and BChE inhibitor, and a non-competitive BACE1 inhibitor, with IC50s of 1.07, 6.03 and 8.55 μM, respectively.

ML352 is a noncompetitive inhibitor of the presynaptic choline transporter.

Isolated from the flower extract of Mentha arvensis, Linarin is a novel and potent acetylcholinesterase inhibitor of acetylcholinesterase (AChE).

Rivastigmine, also known as ENA-713 and SDZ-ENA 713, is a reversible cholinesterase inhibitor with IC50 of 5.5 μM.

Corynoline is a novel and potent AChE inhibitor.

Dehydronuciferine is a novel and potent acetylcholinesterase (AChE) inhibitor.

Epiberberine is a natural anticancer alkaloid isolated from Coptis chinensis with the potential for the treatment of diabetic disease.