2-Hydroxyflutamide (Hydroxyniphtholide), a metabolite of flutamide, is an androgen receptor antagonist potentially for the treatment of prostate cancer.

L-765314 (L-765,314) is a novel, potent and selective α1b adrenergic receptor antagonist with Kis of 5.4 nM and 2.0 nM for rat and human α1b adrenergic receptor, respectively.

Dronedarone (formerly SR-33589; D-03914; S-7529; D-4689; W-3083; RL-01735; Multaq) is a non-iodinated amiodarone analog and a Class III antiarrhythmic as well as multi channel blocker approved for the treatment for Atrial fibrillation (AF).

Formoterol maleate is a long-acting β2 agonist (LABA) used in the treatment of asthma and COPD (chronic obstructive pulmonary disease).

Dexmedetomidine (trade name Precedex), the dexter isomer of medetomidine, is a potent and highly selective alpha-2 adrenergic receptor agonist with sedative activities.

Metoprolol Tartrate (CGP2175E; CGP-2175E; Lanoc; Lopressor; Metomerck; Metop; Selopral; Ritmolol), the tartrate salt of Metoprolol, is a potent and cardioselective β1 receptor blocker with antihypertensive effects.

Oxprenolol HCl (Ba-39089 hydrochloride) is a novel and potent beta blocker with intrinsic sympathomimetic activity.

Brimonidine (UK 14304 and AGN190342) is a highly potent and selective α-adrenergic receptor agonist with EC50 of 0.45 nM for the α2A adrenoreceptor, and used to treat open-angle glaucoma or ocular hypertension.

Metoprolol Succinate (Toprol XL) is a potent and cardioselective β1 receptor blocker medication, which is used to treat hypertension and heart failure.

Maprotiline HCl (Psymion; Ludiomil), the hydrochloride salt of Maprotiline which is a tetracyclic antidepressant, is a selective noradrenalin reuptake inhibitor that has been approved for the treatment of depression.