CCG-63808

This product is for research use only, not for human use. We do not sell to patients.

CCG-63808
For small sizes, please check our retail website as below: www.invivochem.com
Size Price Stock
250mg$830To Be Confirmed
500mg$1140To Be Confirmed
1g$1710To Be Confirmed

Cat #: V4958 CAS #: 620113-73-7 Purity ≥ 98%

Description: CCG-63808 is a novel, potent and reversible inhibitor of regulator of G-protein signaling (RGS) proteins with IC50 value of 1.4 μM for RGS4.

References: Levi L. Blazer et al.Reversible, Allosteric Small-Molecule Inhibitors of Regulator of G Protein Signaling Proteins. Molecular Pharmacology September 2010 vol.78 no.3 524-533

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Product Promise

Promise
Molecular Weight (MW)454.48
Molecular FormulaC25H15FN4O2S
CAS No.620113-73-7
Storage-20℃ for 3 years in powder formr
-80℃ for 2 years in solvent
Preparing Stock Solutions
Solvent volume to be added Mass (the weight of a compound)
Mother liquor concentration 1mg5mg10mg20mg
1mM2.2003 mL11.0016 mL22.0032 mL44.0063 mL
5mM0.4401 mL2.2003 mL4.4006 mL8.8013 mL
10mM0.2200 mL1.1002 mL2.2003 mL4.4006 mL
20mM0.1100 mL0.5501 mL1.1002 mL2.2003 mL
Quality Control Documentation
The molarity calculator equation
Mass(g) = Concentration(mol/L) × Volume(L) × Molecular Weight(g/mol)
Mass
=
Concentration
×
Volume
×
Molecular Weight*
The dilution calculator equation
Concentration(start) × Volume(start) = Concentration(final) × Volume(final)

This equation is commonly abbreviated as: C1 V1 = C2 V2

Concentration(start)
C1
×
Volume(start)
V1
=
Concentration(final)
C2
×
Volume(final)
V2
Step One: Enter information below
Dosage mg/kg Average weight of animals g Dosing volume per animal µL Number of animals
Step Two: Enter the in vivo formulation
%DMSO + % + %Tween 80 + %ddH2O

Calculation Results:
Working concentration: mg/ml;
Method for preparing DMSO master liquid: mg drug pre-dissolved in µL DMSO(Master liquid concentration mg/mL) ,Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.
Method for preparing in vivo formulation: Take µL DMSO master liquid, next add µL PEG300, mix and clarify, next add µL Tween 80,mix and clarify, next add µL ddH2O,mix and clarify.
Note:
  • (1) Please be sure that the solution is clear before the addition of next solvent. Dissolution methods like vortex, ultrasound or warming and heat may be used to aid dissolving.
  • (2) Be sure to add the solvent(s) in order.