This product is for research use only, not for human use. We do not sell to patients.
| Size | Price | Stock |
|---|---|---|
| 5mg | $150 | 3-6 Days |
| 10mg | $250 | 3-6 Days |
| 25mg | $450 | 3-6 Days |
| 50mg | $750 | 3-6 Days |
: Cat #: V17742 CAS #: 1404095-34-6 Purity ≥ 98%
Description: CCT-244747 is a novel, potent, highly selective and orally bioavailable ATP-competitive CHK1 inhibitor (IC50 = 7.7 nM) with potential anticancer activity. CCT244747 inhibited cellular CHK1 activity (IC(50) 29-170 nmol/L), significantly enhanced the cytotoxicity of several anticancer drugs, and abrogated drug-induced S and G(2) arrest in multiple tumor cell lines. CCT244747 represents the first structural disclosure of a highly selective, orally bioavailable CHK1 inhibitor and warrants further evaluation alone or combined with genotoxic anticancer therapies.
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This equation is commonly abbreviated as: C1 V1 = C2 V2
- (1) Please be sure that the solution is clear before the addition of next solvent. Dissolution methods like vortex, ultrasound or warming and heat may be used to aid dissolving.
- (2) Be sure to add the solvent(s) in order.